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Gremlin

Gremlin Informations sur la molécule

Nom anglaisGremlin-1Nombre de médicaments commercialisés0
Nombre de médicaments cliniques2Alias de la cibleCell proliferation-inducing gene 2 protein,Cysteine knot superfamily 1, BMP antagonist 1,DAN domain family member 2,Down-regulated in Mos-transformed cells protein,Increased in high glucose protein 2,IHG-2,CKTSF1B1,DAND2,DRM
Phase de R&D la plus avancéePhase 2 Clinical
Nom anglaisGremlin-1
Alias de la cibleCell proliferation-inducing gene 2 protein,Cysteine knot superfamily 1, BMP antagonist 1,DAN domain family member 2,Down-regulated in Mos-transformed cells protein,Increased in high glucose protein 2,IHG-2,CKTSF1B1,DAND2,DRM
Nombre de médicaments commercialisés0
Nombre de médicaments cliniques2
Phase de R&D la plus avancéePhase 2 Clinical

Gremlin Liste de produits

  • Attribut

    Protein (2)

  • Bibliothèque de produits

    En ligne (2)

  • Espèces

    Human (2)

  • Étiquette

    His Tag (1)Fc Tag (1)

  • Marqueur

    Unconjugated (2)

Numéro de produitEspècesSystème d'expressionDescription du produitStructure protéiquePuretéCaractéristiquesPré-commande/Commande
GR1-H5254
Human
HEK293
Human Gremlin / GREM1 Protein, Fc Tag
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GR1-H52H3
Human
HEK293
Human Gremlin / GREM1 Protein, His Tag
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Quantité totale2
  • 1

GremlinContexte de la molécule

Gremlin is also known as Cysteine knot superfamily 1, BMP antagonist 1 (CKTSF1B1), DAN domain family member 2 (DAND2), Down-regulated in Mos-transformed cells protein (DRM), Increased in high glucose protein 2 (IHG-2), Cell proliferation-inducing gene 2 protein (PIG2) or Gremlin-1 (GREM1), which is highly expressed in small intestine, fetal brain and colon. Gremlin / GREM-1 interacts with SLIT1 and SLIT2 in a glycosylation-dependent manner. Gremlin may play an important role during carcinogenesis and metanephric kidney organogenesis, as a BMP antagonist required for early limb outgrowth and patterning in maintaining the FGF4-SHH feedback loop. Gremlin down-regulates the BMP4 signaling in a dose-dependent manner and acts as inhibitor of monocyte chemotaxis.

GremlinAlias de la molécule

GREM1,CKTSF1B1,DAND2,DRM,PIG2

Informations sur les médicaments cliniques

Nom anglaisCode de recherchePhase de R&DEntrepriseIndicationEssai clinique
TST-003TST-003Phase 2 ClinicalMabspace Biomedicine (Suzhou) Co LtdSolid tumours; Neoplasms; Colorectal Neoplasms; Neoplasm Metastasis
Details
GinisortamabUCB-6114Phase 2 ClinicalUcb Biopharma SrlSolid tumours
Details
  • Liste de produits
  • Informations sur les médicaments cliniques